MgSO4

COc1ccc(C2C(=O)CCc3ccccc32)cc1
Reaction #41960
1-(4-methoxyphenyl)-3,4-dihydro-1H-naphthalene-2-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=C1CCc2ccccc2C1c1ccc2c(c1)OCO2
Reaction #41961
1-benzo[1,3]dioxole-5-yl-3,4-dihydro-1H-naphthalene-2-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1ccc2c(c1)CCC(=O)C2c1ccccc1
Reaction #41962
6-methoxy-1-phenyl-3,4-dihydro-1H-naphthalene-2-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=C1CCc2cc3c(cc2C1c1ccccc1)OCO3
Reaction #41963
5-phenyl-7,8-dihydro-5H-naphtho[2,3-d][1,3]dioxole-6-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CC(C)(C)OC(=O)N[C@@H](Cc1cc(F)cc(F)c1)[C@H](O)CNCc1ccc[nH]1
Reaction #42596
tert-butyl (1S,2R)-1-(3,5-difluorobenzyl)-2-hydroxy-3-[(1H-pyrrol-2-ylmethyl)amino]propylcarbamate
收率 62.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Cc1n[nH]c2ccc3c(=O)c(-c4ccc(Cl)cc4)c(C(C)C)oc3c12
Reaction #42776
product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CC(C)c1oc2c(ccc3[nH]ncc32)c(=O)c1-c1ccc(Cl)cc1
Reaction #42778
3-(4-Chlorophenyl)-2-isopropyl-7H-pyrano[2,3-e]indazol-4-one
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1cc(OC)c2c(CNC(=O)OC(C)(C)C)ncc(Nc3nc(C)cs3)c2c1
Reaction #42926
[6,8-dimethoxy-4-(4-methyl-thiazol-2-ylamino)isoquinolin-1-ylmethyl]carbamic acid tert-butyl ester
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCOC(=O)c1csc(Nc2cnc(CNC(=O)OC(C)(C)C)c3c(OC)cc(OC)cc23)n1
Reaction #42928
2-[1-(tert-butoxycarbonylamino-methyl)-6,8-dimethoxy-isoquinolin-4-ylamino]thiazole-4-carboxylic acid ethyl ester
收率 42.1%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1cc2c(Nc3nc(-c4ccccc4)cs3)cnc(CNC(=O)OC(C)(C)C)c2cc1OC
Reaction #42945
[6,7-dimethoxy-4-(4-phenyl-thiazol-2-ylamino)isoquinolin-1-ylmethyl]carbamic acid tert-butyl ester
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1cc2c(Nc3nc(C)cs3)cnc(CNC(=O)OC(C)(C)C)c2cc1OC
Reaction #42947
[6,7-dimethoxy-4-(4-methyl-thiazol-2-ylamino)isoquinolin-1-ylmethyl]carbamic acid tert-butyl ester
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCOC(=O)c1csc(Nc2cnc(CNC(=O)OC(C)(C)C)c3cc(OC)c(OC)cc23)n1
Reaction #42949
2-[1-(tert-butoxycarbonylamino-methyl)-6,7-dimethoxy-isoquinolin-4-ylamino]thiazole-4-carboxylic acid ethyl ester
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CCOC(=O)C(C)=NNC
Reaction #44233
desired product
收率 94.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COC(=O)[C@@H](/N=C/c1cccc(Br)n1)C(C)C
Reaction #45391
(S)-2-{[1-(6-Bromo-pyridin-2-yl)-meth-(E)-ylidene]-amino}-3-methyl-butyric acid methyl ester
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
COc1c(F)cc(C)cc1C(=NO)C(N)=O
Reaction #45565
compound
收率 10.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
O=S(=O)(CC1CNC1)c1ccccc1
Reaction #46339
3-(phenylsulfonylmethyl)azetidine
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
C[C@H](N[C@H](CO)COCc1ccccc1)C(OCC(C)(C)C)OCC(C)(C)C
Reaction #48682
title compounds
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
CC(C)[Si](OC(=CCl)c1ncccn1)(C(C)C)C(C)C
Reaction #51973
product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2005_02
CC(C)(C)OC(=O)CN1C(c2ccccc2)COC1C(c1ccccc1)c1ccccc1
Reaction #53952
tert-butyl (2-benzhydryl-4-phenyl-oxazolidin-3-yl)-acetate
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2005_02
CC(C)(C)OC(=O)CN1C(C(c2ccccc2)c2ccccc2)OC[C@H]1c1ccccc1
Reaction #53960
tert-butyl ((4R)-2-benzhydryl-4-phenyl-oxazolidin-3-yl)-acetate
收率 114.1%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2005_02