4-borono-2-fluorobenzoic acid

O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #84065
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_09
Nc1n[nH]c2cc(-c3ccc(C(=O)O)c(F)c3)nc(-c3ccc(Oc4ccccc4)cc3)c12
Reaction #168256
desired product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09
CCS(=O)(=O)c1ccc(-c2ccc(C(=O)O)c(F)c2)cn1
Reaction #402717
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (8/10)
—
Reaction #494050
solid
Rendement 19.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_06
CS(=O)(=O)c1cccc(CNC(=O)c2ccc(B(O)O)cc2F)c1
Reaction #682973
3-fluoro-4-(3-(methylsulfonyl)benzylcarbamoyl)-phenylboronic acid
Rendement 88.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_01
O=C(NC(c1ccccc1)C(F)(F)F)c1ccc(B(O)O)cc1F
Reaction #682974
crude product
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_01
O=C(N[C@@H]1CCCN(S(=O)(=O)c2ccccc2F)C1)c1ccc(B(O)O)cc1F
Reaction #682977
(R)-3-fluoro-4-(1-(2-fluorophenylsulfonyl)piperidin-3-ylcarbamoyl)phenylboronic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_01
O=C(NC(c1ccccc1)C(F)F)c1ccc(B(O)O)cc1F
Reaction #682979
4-(2,2-difluoro-1-phenylethylcarbamoyl)-3-fluorophenylboronic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_01
Nc1ncc(C2CCOCC2)cc1-c1ccc(C(=O)O)c(F)c1
Reaction #683244
4-(2-Amino-5-(tetrahydro-2H-pyran-4-yl)pyridin-3-yl)-2-fluorobenzoic acid
Rendement 137.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_01
O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #716041
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_04
O=C(c1ccc(B(O)O)cc1F)N1CCOCC1
Reaction #719655
crude compound
Rendement 87.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_04
O=C(c1ccc(B(O)O)cc1F)N1CCC(F)(F)C1
Reaction #775706
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (3/10)
O=C(c1ccc(B(O)O)cc1F)N1CCOCC1
Reaction #1140298
crude compound
Rendement 87.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2016_07
O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #1497747
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_12
O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #1559824
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2015_04
O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #1594520
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2015_12
O=C(O)c1ccc(-c2ccc3cc(O)ccc3n2)cc1F
Reaction #1714797
2-fluoro-4-(6-hydroxyquinolin-2-yl)benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_07
C[C@@H]1CCCN1C[C@@H]1CCCN1C(=O)c1ccc(-c2ccc(C(=O)C3CC3)cc2)cc1F
Reaction #1764380
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_08
CC1(C)OB(c2ccc(C(=O)O)c(F)c2)OC1(C)C
Reaction #1764381
2-Fluoro-4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_08
CCS(=O)(=O)c1ccc(-c2ccc(C(=O)O)c(F)c2)cn1
Reaction #1764382
4-(6-Ethanesulfonyl-pyridin-3-yl)-2-fluoro-benzoic acid
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_08
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