5-fluoro-1H-indole-2-carboxylic acid

O=C(NCCCO)c1cc2cc(F)ccc2[nH]1
Reaction #58061
5-fluoro-1H-indole-2-carboxylic acid (3-hydroxy-propyl)-amide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2008_09
Nc1ccc(OCc2ccccc2)c(CO)c1
Reaction #60606
4-benzyloxy-3-hydroxymethylaniline
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2008_09
CC(C)(C)C(NC(=O)c1cc2cc(F)ccc2[nH]1)C(=O)N1CC2CC1CN2C(=O)c1ccc(-c2ccccc2)cn1
Reaction #177467
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)
COC(=O)C1CCC(NC(=O)c2cc3cc(F)ccc3[nH]2)C(NC(=O)c2nc3c(s2)CN(C)CC3)C1
Reaction #178101
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)
CCc1cc(C(=O)c2ccccc2Cl)c(-n2c(C)nnc2CNC(=O)c2cc3cc(F)ccc3[nH]2)s1
Reaction #195744
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)
O=C(Cl)c1cc2cc(F)ccc2[nH]1
Reaction #226479
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)
O=C(c1cc2cc(F)ccc2[nH]1)N1CCN(c2ccccn2)CC1
Reaction #237699
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)
O=C(NC1CCN(CCn2c(=O)cnc3ccc(F)cc32)CC1)c1cc2cc(F)ccc2[nH]1
Reaction #247671
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (9/10)
O=C(NC(Cc1ccc(F)cc1)C(=O)N1CCC(O)CC1)c1cc2cc(F)ccc2[nH]1
Reaction #294822
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (6/10)
O=C(NC1CCN(CCn2c(=O)cnc3ccc(F)cc32)CC1)c1cc2cc(F)ccc2[nH]1
Reaction #342525
title compound
Ausbeute 79.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_01
Nc1ccc(OCc2ccccc2)c(CO)c1
Reaction #502224
4-benzyloxy-3-hydroxymethylaniline
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2012_01
COC(=O)[C@@H]1CC[C@H](NC(=O)c2cc3cc(F)ccc3[nH]2)[C@H](NC(=O)c2nc3c(s2)CN(C)CC3)C1.Cl
Reaction #546764
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2007_03
Nc1ccc(OCc2ccccc2)c(CO)c1
Reaction #587612
4-benzyloxy-3-hydroxymethylaniline
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_08
COC(=O)[C@@H]1CC[C@H](NC(=O)c2cc3cc(F)ccc3[nH]2)[C@H](NC(=O)c2nc3c(s2)CN(C)CC3)C1.Cl
Reaction #633711
title compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_05
CC1(C)Cc2ccc(C#N)cc2[C@@H]1NC(=O)c1cc2cc(F)ccc2[nH]1
Reaction #636633
desired title product
Ausbeute 76.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_05
O=C(N[C@@H](Cc1ccccc1)C(=O)N1CCC(O)CC1)c1cc2cc(F)ccc2[nH]1
Reaction #738296
5-Fluoro-1H-indole-2-carboxylic acid [(1S)-benzyl-2-(4-hydroxy-piperidin-1-yl)-2-oxo-ethyl]-amide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2001_08
O=C(N[C@@H](Cc1ccc(F)cc1)C(=O)N1CCOCC1)c1cc2cc(F)ccc2[nH]1
Reaction #738298
5-Fluoro-1H-indole-2-carboxylic acid [(1S)-(4-fluoro-benzyl)-2-morpholin-4-yl-2-oxo-ethyl]-amide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2001_08
O=C(N[C@@H](Cc1ccc(F)cc1)C(=O)N1CCC(O)CC1)c1cc2cc(F)ccc2[nH]1
Reaction #738326
5-Fluoro-1H-indole-2-carboxylic acid [(1S)-(4-fluoro-benzyl)-2-(4-hydroxy-piperidin-1-yl)-2-oxo-ethyl]-amide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2001_08
O=C(c1cc2cc(F)ccc2[nH]1)N1CCCN(c2ccccn2)CC1
Reaction #757675
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (3/10)
O=C(c1cc2cc(F)ccc2[nH]1)N1CC2CC1CN2c1ccccn1
Reaction #762530
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (3/10)
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