DEAD toluene
Reaction #49376
4-[2-(dimethylamino)ethoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 53.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49377
(3-(tert-butoxycarbonylamino)propoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 88.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49378
4-[3-(tert-butyldimethylsilyloxy)propoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 53.4%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49399
4-[3-(tert-butoxycarbonylamino)propoxy]-7-[1-(tert-butoxycarbonyl)-5-formylindol-2-yl]isoindolinone
Ausbeute 99.1%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49402
4-benzyloxy-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 73.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49403
4-(2-isopropoxyethoxy)-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 59.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49404
4-[3-(dimethylamino)propoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 39.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49405
4-[3-(4-methylpiperazin-1-yl)propoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidinomethyl)indol-2-yl]isoindolinone
Ausbeute 58.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #49592
4-chloro-5-[3-(tert-butyldimethylsiloxy)propoxy]-7-[1-(tert-butoxycarbonyl)-5-(piperidin-1-ylmethyl)indol-2-yl]isoindolinone
Ausbeute 64.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Reaction #435921
compound
Ausbeute 67.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2007_02
Reaction #689364
desired compound
Ausbeute 67.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_03
Reaction #1261174
compound
Ausbeute 67.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_11
Reaction #1606902
4-[2-(4-iodophenoxy)ethyl]morpholine
Ausbeute 93.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2015_07
Reaction #2508176
4-(2-aminoethyl)pyridine-2-carbonitrile dihydrochloride
Ausbeute 55.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2011_06