反应 #77141

ord-7585679821ee45419a3aa02636c4d30c

反应方程式

COc1cc2c(cc1O)C(Cc1ccc(OC)c(OC)c1)N(CC(=O)NC1CCc3ccccc31)CC2
2-[1-(3,4-dimethoxy-benzyl)-7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-N-(indan-1-yl)-acetamide
Clc1cnccn1
2-chloro-pyrazine
COc1ccc(CC2c3cc(Oc4cnccn4)c(OC)cc3CCN2CC(=O)NC2CCc3ccccc32)cc1OC
2-[1-(3,4-dimethoxy-benzyl)-6-methoxy-7-(pyrazin-2-yloxy)-3,4-dihydro-1H-isoquinolin-2-yl]-N-(indan-1-yl)-acetamide

反应条件

详细条件
See reaction.notes.procedure_details.

实验过程

prepared by reaction of 2-[1-(3,4-dimethoxy-benzyl)-7-hydroxy-6-methoxy-3,4-dihydro-1H-isoquinolin-2-yl]-N-(indan-1-yl)-acetamide with 2-chloro-pyrazine

来源

DOI: 10.6084/m9.figshare.5104873.v1专利: US06703392B2uspto-grants-2004_03