反应 #1797537

ord-95ca348ed32a464eb7f38d05c306dc7d

反应方程式

O=C(NC1C2CC3CC(C2)CC1C3)c1cnn(-c2ccccc2)c1Cl
5-chloro-1-phenyl-1H-pyrazole-4-carboxylic acid adamantan-2-ylamide
O=C(NC1C2CC3CC(C2)CC1C3)c1cnn(-c2ccccc2)c1Cl
Intermediate 3
O=C(NC1C2CC3CC(C2)CC1C3)c1cnn(-c2ccccc2)c1Cl
5-chloro-1-phenyl-1H-pyrazole-4-carboxylic acid adamantan-2-ylamide
OC[C@@H]1CCCN1
L-prolinol
O=C(NC1C2CC3CC(C2)CC1C3)c1cnn(-c2ccccc2)c1N1CCC[C@H]1CO
5-((S)-2-Hydroxymethyl-pyrrolidin-1-y1)-1-phenyl- 1H-pyrazole-4-carboxylic acid adamantan-2-ylamide

反应条件

详细条件
See reaction.notes.procedure_details.

实验过程

5-((S)-2-Hydroxymethyl-pyrrolidin-1-y1)-1-phenyl- 1H-pyrazole-4-carboxylic acid adamantan-2-ylamide was prepared using Procedure A from 5-chloro-1-phenyl-1H-pyrazole-4-carboxylic acid adamantan-2-ylamide (Intermediate 3) and L-prolinol. Mass spectrum (ES) MH+=421.

来源

DOI: 10.6084/m9.figshare.5104873.v1专利: US07790711B2uspto-grants-2010_09