参与 66 个反应

6084

Cc1ccccc1NC(=O)c1ccc(C(=O)N2Cc3cccn3Cc3ccccc32)cc1
Reaction #3673
white crystals
收率 54.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1998_03
Cc1cccc(NC(=O)c2ccc(C(=O)N3Cc4cccn4Cc4ccccc43)cc2)c1C
Reaction #3674
crystals
收率 25.4%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1998_03
COCCNC(=O)c1cnc(CNC(=O)OC(C)(C)C)c2cc(OC)c(OC)cc12
Reaction #42933
[6,7-dimethoxy-4-(2-methoxy-ethylcarbamoyl)-isoquinolin-1-ylmethyl]-carbamic acid tert-butyl ester
收率 49.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2010_06
Cc1ccccc1NC(=O)c1ccc(C(=O)N2Cc3cccn3Cc3ccccc32)cc1
Reaction #83494
white crystals
收率 54.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04
Cc1cccc(NC(=O)c2ccc(C(=O)N3Cc4cccn4Cc4ccccc43)cc2)c1C
Reaction #83495
crystals
收率 25.4%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04
COc1cc(C(=O)NNC(=O)OC(C)(C)C)ccc1-n1cnc(C)c1
Reaction #158321
title compound
收率 44.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09
CO[C@H]([C@@H](C)C(=O)N[C@@H](Cc1ccccc1)c1nccs1)[C@@H]1CCCN1C(=O)OC(C)(C)C
Reaction #161910
#16
收率 81.1%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_09
O=C1NC(=O)C(c2ccc(NC(=O)c3ccc4c(c3)OCO4)cc2)S1
Reaction #174865
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (2/10)
CC(C)(C)OC(=O)N1C(c2cccnc2)SC[C@H]1C(=O)NCCCN1CCN(C(c2ccccc2)c2ccccc2)CC1
Reaction #216930
title compound
收率 89.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1995_11
CN(C)C(=O)c1cc(Br)cnc1N
Reaction #328241
title Compound
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-2014_02
Cc1cc(C)c2ncc(NC(=O)c3cc(C(C)(C)C)c(O)c(C(C)(C)C)c3)c(-c3ccccc3Cl)c2c1
Reaction #347037
4-(2-chlorophenyl)-3-(3,5-di-tert-butyl-4-hydroxybenzamido)-6,8-dimethylquinoline
收率 24.2%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1996_06
O=C(C=c1sc2n(c1=O)Cc1ccccc1N=2)NCc1ccccc1
Reaction #367556
N-Benzyl-(3-oxo-5H-thiazolo[2,3-b]quinazolin-2(3H)-ylidene)acetamide
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1986_05
Cc1cccc(NC(=O)c2ccc(C(=O)N3Cc4cccn4Cc4ccccc43)cc2)c1C
Reaction #403689
DOI: 10.1039/C8SC04228DTraining data from https://doi.org/10.1039/C8SC04228D (8/10)
CC[C@H](C)[C@H](NC(=O)[C@@H](N)CCCCN)C(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)[C@H](O)[C@@H]1O.Cl.Cl
Reaction #417018
5'-O-(N-Lysylisoleucyl)-5-fluorouridine dihydrochloride
DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1990_01
CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CCCCNC(=O)OCc1ccccc1)NC(=O)OCc1ccccc1)C(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)[C@H](O)[C@@H]1O
Reaction #417019
5'-O-[N-{N-(Nα,Nε -di benzyloxycarbonyllysyl)alanyl}isoleucyl]-5-fluorouridine
收率 45.9%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1990_01
CC[C@H](C)[C@H](NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)C(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)[C@H](O)[C@@H]1O
Reaction #417021
5'-O-[N-{(N-benzyloxycarbonylphenylalanyl)alanyl}isoleucyl]-5-fluorouridine
收率 35.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1990_01
CC[C@H](C)[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](C)NC(=O)[C@H](CCCCNC(=O)OCc1ccccc1)NC(=O)OCc1ccccc1)C(=O)OC[C@H]1O[C@@H](n2cc(F)c(=O)[nH]c2=O)[C@H](O)[C@@H]1O
Reaction #417022
5'-O-[N-[N-{N-(Nα,Nε -dibenzyloxycarbonyllysyl)alanyl}phenylalanyl]isoleucyl]-5-fluorouridine
收率 52.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1990_01
Cc1ccccc1NC(=O)c1ccc(C(=O)N2Cc3cccn3Cc3ccccc32)cc1
Reaction #527198
white crystals
收率 54.6%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1996_05
Cc1cccc(NC(=O)c2ccc(C(=O)N3Cc4cccn4Cc4ccccc43)cc2)c1C
Reaction #527199
crystals
收率 25.4%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1996_05
COc1ccc(C(=O)N2CCC[C@H]2C(OC)OC)cc1
Reaction #554331
title compound
收率 65.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1992_10
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