6-fluoro-3-(4-piperidinyl)-1,2-benzisoxazole

COc1ccccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1.O=C(O)/C=C/C(=O)O

Reaction #83852

6-fluoro-3-[1-[3-(2-methoxyphenoxy)-propyl]-4-piperidinyl]-1,2-benzisoxazole fumarate

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1ccc(C2(C=O)C=CC=CC2)cc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83853

1-[3-[3-[4-(6- fluoro-1,2-benzisoxa zol-3-yl)-1-piperidinyl]propoxy]-4-methoxyphenyl]-phenylmethanone

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C#N)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83861

4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3-methoxybenzonitrile

收率 68.2%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CC(=O)c1cc(Br)c(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c(Br)c1

Reaction #83862

1-[3,5-dibromo-4-[3-[4-(6-fluoro-1,2- benzisoxazol-3-yl)-1-piperidinyl]propoxy]-phenyl]ethanone

收率 58.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

Fc1ccc2c(C3CCN(CCCOc4ccccc4)CC3)noc2c1

Reaction #83863

6-fluoro-3-[1-(3-phenoxypropyl)-4-piperidinyl]-1,2-benzisoxazole

收率 47.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C(=O)C(F)(F)F)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83864

1-[4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]-propoxy]-3-methoxyphenyl]-2,2,2-trifluoro-ethanone

收率 56.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CSc1cc(C(C)=O)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83865

1-[4-[3-[4-(6-fluoro-1,2-benzoisoxazol-3-yl]-1-piperidinyl]propoxy]-3-methylmercaptophenyl]ethanone

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C2(C=O)C=CC=CC2)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83867

off-white solid

收率 87.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CCCC(=O)Cc1ccc(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c(OC)c1

Reaction #83868

1-[4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl )-1-piperidinyl]propoxy]-3-methoxyphenyl]-pentanone

收率 68.7%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(CC(C)=O)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83869

1-[4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3-methoxyphenyl]propanone

收率 31.8%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C(N)=O)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83870

4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3-methoxybenzamide

收率 64.3%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CNc1cc(C(C)=O)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83871

1-[4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3-(methylamino)phenyl]ethanone

收率 47.9%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CC(=O)Nc1cccc(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c1.CC(=O)Nc1cccc(OCCCN2CCC(c3noc4cc(F)ccc34)CC2)c1.O=C(O)/C=C/C(=O)O

Reaction #83884

N-[3-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]phenyl]acetamide hemifumarate

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C(=O)N(C)C)ccc1OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83888

N,N-dimethyl-4-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propoxy]-3methoxybenzamide

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

OCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83892

6-fluoro-3-[1-(3-hydroxypropyl)-4-piperidinyl]-1,2-benzisoxazole

收率 63.9%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

Fc1ccc2c(C3CCN(CC4COc5ccccc5O4)CC3)noc2c1

Reaction #83893

2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]methyl-1,4-benzodioxan

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

CC(=O)c1ccc2c(c1)oc(=O)n2CCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83897

N-[3-[4-(6-fluoro-1,2-benzisoxazol-3yl)-1-piperidinyl]propyl]-6-acetyl-2-benzoxazolinone

收率 31.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

O=C1c2ccccc2C(=O)N1CCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83898

N-[3-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]propyl]phthalimide

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

COc1cc(C(C)=O)ccc1SCCCN1CCC(c2noc3cc(F)ccc23)CC1

Reaction #83904

light brown oil

收率 113.0%DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

$CCCC(c1ccccc1OC)N1CCC(c2noc3cc(F)ccc23)CC1.O=C(O)/C=C\C(=O)O$

Reaction #83905

4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-(2'-methoxyphenyl)butylpiperidine maleate

DOI: 10.6084/m9.figshare.5104873.v1uspto-grants-1997_04

第 1 页下一页