Реакция #58455

Уравнение реакции

(RS)-2-carboxymethyl-piperidine-1-carboxylic acid tert butyl ester

2-bromo-4′-fluoroacetophenone

→

title compound

Выход 96.9%

(RS)-2-[2-(4-Fluoro-phenyl)-2-oxo-ethoxycarbonylmethyl]-piperidine-1-carboxylic tert butyl ester

Выход 96.9%

Условия реакции

Методика

The title compound (3.83 g) was prepared from (RS)-2-carboxymethyl-piperidine-1-carboxylic acid tert butyl ester (2.54 g) and 2-bromo-4′-fluoroacetophenone (2.26 g) according to the method of description 36.

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