Реакция #467733

Уравнение реакции

naphthalene-2-boronic acid

1-phenoxycarbonyl-2-ethyl-4-trifluoromethanesulfonyloxy-1,2,3,6-tetrahydropyridine

→

desired compound

Выход 75.3%

1-phenoxycarbonyl-2-ethyl-4-(naphth-2-yl)-1,2,3,6-tetrahydropyridine

Выход 75.3%

Условия реакции

Методика

Beginning with 3.62 gm (21.1 mMol) naphthalene-2-boronic acid and 5.70 gm (15.0 mMol) 1-phenoxycarbonyl-2-ethyl-4-trifluoromethanesulfonyloxy-1,2,3,6-tetrahydropyridine, 4.04 gm (75%) of the desired compound were prepared substantially as described in EXAMPLE 11.

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