Реакция #46563

Уравнение реакции

( c )

5-bromo-2-(methoxycarbonylmethyl)aminopyridine

4-chloro-1-methyl-1H-indole-3-carboxaldehyde

1,3-dimethyl-1H-indole-2-carboxaldehyde

→

title compound

Выход 78.0%

4-Chloro-1-methyl-3-(methylaminomethyl)-1H-indole

Выход 78.0%

Условия реакции

Методика

According to the procedure of Preparation 13 (c), except substituting 4-chloro-1-methyl-1H-indole-3-carboxaldehyde for the 1,3-dimethyl-1H-indole-2-carboxaldehyde, the title compound (1.75 g, 78%) was obtained as a yellow solid: MS (ES) m/e 209.0 (M+H)+.

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