Реакция #426862

Уравнение реакции

2-(7-(2-methoxyethoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)quinolin-8-yl trifluoromethane sulfonate

tert-butyl piperidin-4-ylmethylcarbamate

tert-butyl piperazine-1-carboxylate

→

tert-butyl(1-(2-formylquinolin-8-yl)piperidin-4-yl)methylcarbamate

Условия реакции

Обработка

1. 1
   ДругоеPrepared

Методика

Prepared as described in Example 1, Step H, substituting 8-bromoquinoline-2-carbaldehyde for 2-(7-(2-methoxyethoxy)-[1,2,4]triazolo[4,3-a]pyridin-3-yl)quinolin-8-yl trifluoromethane sulfonate, and tert-butyl piperidin-4-ylmethylcarbamate for tert-butyl piperazine-1-carboxylate.

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