Реакция #41347

ord-fa9827dbfe56436cbb15b5c008b0313e

Условия реакции

Подробные условия
See reaction.notes.procedure_details.

Обработка

  1. 1
    ДругоеPrepared

Методика

Prepared as described in Example 1 using (1R,2S)-1-[1-(4-fluorophenyl)-6-methyl-indazol-5-yl]oxy-1-phenyl-propan-2-amine (50 mg, 0.13 mmol) and pivaloyl chloride (0.065 mL, 0.53 mmol). Yield 53 mg (87%).

Источник

DOI: 10.6084/m9.figshare.5104873.v1Патент: US07728030B2uspto-grants-2010_06