Реакция #2275763

Уравнение реакции

(4-oxo-cyclohexyl)-carbamic acid tert-butyl ester

N-(azetidin-3-ylcarbamoylmethyl)-3-trifluoromethyl-benzamide

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title compounds

{4-{3-[2-(3-Trifluoromethyl-benzoylamino)-acetylamino]-azetidin-1-yl}-cyclohexyl)-carbamic acid tert-butyl ester

Условия реакции

Методика

The title compounds were prepared as white solids from the reductive amination of (4-oxo-cyclohexyl)-carbamic acid tert-butyl ester (Asta) and N-(azetidin-3-ylcarbamoylmethyl)-3-trifluoromethyl-benzamide (as prepared in Example 2 Step C) using the procedure described in Step D of Example 1.

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