Реакция #1683000

ord-2a93b5e8f23c45289e0aa8ad7305490f

Уравнение реакции

COc1cc2ncc(C#N)c(Cl)c2cc1OC
4-chloro-6,7-dimethoxy-3-quinolinecarbonitrile
Cn1ccnc1Sc1ccc(N)cc1Cl
3-chloro-4-(1-methyl-2-imidazolylthio)aniline
COc1cc2ncc(C#N)c(Nc3ccc(Sc4nccn4C)c(Cl)c3)c2cc1OC
title compound
COc1cc2ncc(C#N)c(Nc3ccc(Sc4nccn4C)c(Cl)c3)c2cc1OC
4-[3-Chloro-4-(1-methyl-2-imidazolylthio)phenylamino]-6,7-dimethoxy-3-quinolinecarbonitrile

Условия реакции

Подробные условия
See reaction.notes.procedure_details.

Методика

In the manner of Example 141 reaction of 4-chloro-6,7-dimethoxy-3-quinolinecarbonitrile with 3-chloro-4-(1-methyl-2-imidazolylthio)aniline (WO-9615118) gave the title compound as a white solid, mp 302-307° C.

Источник

DOI: 10.6084/m9.figshare.5104873.v1Патент: US06288082B1uspto-grants-2001_09