Реакция #1563958

ord-f0087ca7544940939a7e73010b3825e8

Условия реакции

Подробные условия
See reaction.notes.procedure_details.

Обработка

  1. 1
    Другоеto afford as yellow solid

Методика

The title compound (Int-72) was prepared by the method similar to that for Int-84 using (R)-2-(2,5-difluorophenyl)-4,4-difluoropyrrolidine hydrochloride and Ethyl 5-bromopyrazolo[1,5-a]pyridine-3-carboxylate to afford as yellow solid. LCMS (ESI): m/z 408.1 (M+H).

Источник

DOI: 10.6084/m9.figshare.5104873.v1Патент: US09402833B2uspto-grants-2016_08