반응 #94060

ord-718f89131b9946e48179fab1305fef8b

반응 방정식

O=C1c2ccccc2CCc2c1nc1c(cnn1Cc1ccccc1)c2O
product
O=C1c2ccccc2CCc2c1nc1c(cnn1Cc1ccccc1)c2O
1-benzyl-5,6-dihydro-4-hydroxybenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-11(1H)one
O=P(Br)(Br)Br
phosphorus oxybromide
O=P(Cl)(Cl)Cl
phosphorus oxychloride
O=C1c2ccccc2CCc2c1nc1c(cnn1Cc1ccccc1)c2Br
1-benzyl-4-bromo-5,6-dihydrobenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-11(1H)one

반응 조건

상세 조건
See reaction.notes.procedure_details.

실험 절차

By treating the product of Example 10 according to the procedure of Example 2, but substituting phosphorus oxybromide for the phosphorus oxychloride, 1-benzyl-4-bromo-5,6-dihydrobenzo[5,6]cyclohepta[1,2-b]pyrazolo[4,3-e]pyridin-11(1H)one is obtained.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04128717uspto-grants-1978_12