반응 #84048

ord-0186fe48a824439e807128658024c08c

반응 방정식

Cl.O=C1CN2CCC1CC2
quinuclidin-3-one hydrochloride
C[O-].[Na+]
sodium methoxide
O=C1CN2CCC1CC2
title compound
O=C1CN2CCC1CC2
Quinuclidin-3-one

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    여과The resulting precipitate is filtered off with suction
  2. 2
    농축the filtrate is concentrated in vacuo
  3. 3
    기타The residue is partitioned between chloroform and water
  4. 4
    추출extracted with chloroform
  5. 5
    건조The combined organic phases are dried over sodium sulfate
  6. 6
    농축concentrated in vacuo

실험 절차

100 g (0.62 mol) of quinuclidin-3-one hydrochloride are suspended in 2 l of methanol. At 0° C., a solution of 33.4 g (0.62 mol) of sodium methoxide in 250 ml of methanol is slowly added dropwise. The mixture is stirred at room temperature for 16 h. The resulting precipitate is filtered off with suction, and the filtrate is concentrated in vacuo. The residue is partitioned between chloroform and water and extracted with chloroform. The combined organic phases are dried over sodium sulfate and concentrated in vacuo. 58.8 g (75.9% of theory) of the title compound are obtained.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US09433614B2uspto-grants-2016_09