반응 #78831

ord-9f0654f057744021bbd1ae4e394cd7af

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타After the completion of the reaction
  2. 2
    농축the mixed liquid was concentrated
  3. 3
    기타the residue was chromatographed in a silica gel column with hexane/ethyl acetate (=8/2) as a developing solvent

실험 절차

Into 0.5 ml of ethanol was dissolved tricyclo[4,2,1,03,9]nonane-2-one (13.6 mg, 0.1 mmol). Into this ethanol solution was added the Co (III) (salen) complex (3.7 mg, 5 μmol) having the above formula (XI). Into this solution was added 30% hydrogen peroxide aqueous solution (15 μI, hydrogen peroxide content 0.13 mmol), which was stirred at room temperature for 24 hours. After the completion of the reaction, the mixed liquid was concentrated, and the residue was chromatographed in a silica gel column with hexane/ethyl acetate (=8/2) as a developing solvent, thereby obtaining 2-oxatricyclo[5.2.1.04,10]decane-3-one (4.7 mg, yield 31%) having the above formula (VIII). The enantiomer excess percentage of the product was determined as follows.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US06713435B2uspto-grants-2004_03