반응 #74767

ord-d06799c8e7d2446093d305f30ce0c2ac

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도the mixture was heated on a steam-bath for 0.5 hours
  2. 2
    여과The mixture was filtered
  3. 3
    농축concentrated
  4. 4
    추출extracted with chloroform
  5. 5
    추출the chloroform extract
  6. 6
    기타was evaporated

실험 절차

A solution of sodium nitrite (2.38 g) in water (10 ml) was added dropwise to a mixture of 3-amino-2-hydroxymethylpyridine (4.8 g), aqueous hydrochloric acid (48%, 10 ml) and water (5 ml) stirred at 0°-5°. This solution was added to a hot solution of cuprous chloride (2.5 g) in conc. hydrochloric acid and the mixture was heated on a steam-bath for 0.5 hours, diluted with water and saturated with hydrogen sulphide. The mixture was filtered, concentrated and extracted with chloroform and the chloroform extract was evaporated to give 3-chloro-2-hydroxymethylpyridine (3.7 g) m.p. 42°-44° (from n-pentane).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04173644uspto-grants-1979_11