반응 #656163

ord-cdffc9b431c346c79072bd402f130673

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타gives an oil which

실험 절차

A mixture of 2,2-difluoro-5-methoxy-1-pentanal hydrate (1.57 g, 9.2 mmoles), hydroxylamino hydrochloride (640 mg, 9.2 mmoles), 1N NaOH (9.2 ml), and dioxane (15 ml) is kept for 1 hour at room temperature. After addition of ether and brine, usual extraction gives an oil which according to NMR is the oxime hydrate. Several evaporations with carbon tetrachloride (50° C., 60 mm Hg) afford the oxime (1.4 g) which is purified by chromatography on silica (ethyl acetate/petroleum ether: 20/80, RF: 0.53): 1.05 g (68%).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04730006uspto-grants-1988_03