반응 #65038

ord-5196aa637c7740218f9e817e1b948708

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도at reflux temperature for 18 hours
  2. 2
    기타was removed by filtration
  3. 3
    기타The excess piperidine is removed by simple distillation
  4. 4
    기타the resultant solid residue is recrystallized from ethanol and water
  5. 5
    기타After drying

실험 절차

11-Bromoundecanol (11.00 g., 43.79 mmole) was dissolved in 100 ml. of piperidine and heated at reflux temperature for 18 hours. The reaction mixture was allowed to cool and most of the precipitated piperidine hydrobromide was removed by filtration. The excess piperidine is removed by simple distillation and the resultant solid residue is recrystallized from ethanol and water. After drying, 10.78 g. (96.3% yield) of 1-hydroxy-11-(N-piperidyl)undecane was obtained. m.p. 62°-65° C., 1H-NMR (200 MHz, CDCl3) δ=1.2-1.7 ppm, m, 24H; 2.10, broad s, 1H; 2.20-2.45, m, 6H; 3.63, t, 2H.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05416210uspto-grants-1995_05