반응 #62570

ord-611285cd275a424f86977e849e6ea951

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    여과The white solid was filtered
  2. 2
    세척washed with water
  3. 3
    건조dried in vacuo over P2O5

실험 절차

4-Iodoveratrole (26.0 g, 0.0985M) in acetic acid (25 ml) was treated with bromine (6.5 ml, 0.127M) in acetic acid (30 ml) and stirred at room temperature for one hour. The mixture was diluted with water (300 ml) and treated with sodium bisulfite to discharge the excess bromine. The white solid was filtered, washed with water and dried in vacuo over P2O5 to give 4-bromo-5-iodoveratrole (33.0 g, 95% yield) as a white solid, mp 98°-100° C. (literature: Baker et al., J. Chem. Soc. 3986 (1961), mp 102°-104° C.). NMR (CDCl3) δ 3.83 ppm (s, 6H, (2x) OCH3), 7.06 (s, 1H, ArH), 7.21 (s, 1H, ArH).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04761413uspto-grants-1988_08