반응 #56297

ord-5a172908a35746a1ae556a5be665f22e

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타viscous residue is obtained
  2. 2
    기타The solid is triturated
  3. 3
    여과collected by filtration
  4. 4
    세척washed with ether
  5. 5
    건조dried over phosphorus pentoxide

실험 절차

7β-(t-Butoxycarbonyl)amino-3-[2-(N-carboethoxysulfamoyl)benzoyloxy]methyl-3-cephem-4-carboxylic acid (2.2 g) is dissolved in ice cooled solution of trifuoroacetic acid (20 ml) and the mixture is stirred for 20 minutes. Then trifluoroacetic acid is taken off under reduced pressure and viscous residue is obtained. The residue becomes solid upon addition of ether (50 ml). The solid is triturated, collected by filtration, washed with ether and dried over phosphorus pentoxide. The procedure provides 7β-amino-3-[2-(N-carboethoxysulfamoyl)benzoyloxy]methyl-3-cephem-4-carboxylic acid (1.55 g).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04224441uspto-grants-1980_09