반응 #5604

ord-e8381d73f4f9423dbff70d4f1bb4f249

반응 방정식

Cc1ccccc1
toluene
C1CCNC1
pyrrolidine
CCOC(=O)CBr
ethyl bromoacetate
CCOC(=O)CN1CCCC1
ETHYL 1-PYRROLIDINEACETATE

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도maintaining the temperature below 30° C
  2. 2
    기타to precipitate pyrrolidinium bromide, which
  3. 3
    기타was separated by filtration
  4. 4
    기타The filtrate was evaporated under vacuum
  5. 5
    기타to provide a residue of about 241 g of ethyl 1-pyrrolinidineacetate

실험 절차

To an ice bath-cooled solution of 213.4 g (3 mol) of pyrrolidine in 450 mL of tetrahydrofuran was added dropwise over about 2 hours 250.5 g (1.5 mol) of ethyl bromoacetate, maintaining the temperature below 30° C. To this solution was added 150 mL of toluene to precipitate pyrrolidinium bromide, which was separated by filtration. The filtrate was evaporated under vacuum to provide a residue of about 241 g of ethyl 1-pyrrolinidineacetate.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05244997uspto-grants-1993_09