반응 #54820

ord-e17b2a24b9b4443fb29dd5a58e75c0fb

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    추출extracted with ether (400 ml total)
  2. 2
    세척the extracts washed
  3. 3
    건조dried (MgSO4)
  4. 4
    기타evaporated
  5. 5
    기타The resulting crude solid (2.2 g) is recrystallized from toluene

실험 절차

Sodium hydroxide (0.40 g. of 50% dispersion in mineral oil) is added to 0.61 g. imidazole in 10 ml dimethylformamide and the mixture stirred at room temperature until the evolution of hydrogen is complete. Bromomethyl 2-naphthoyl ketone dimethyl ketal (2.21 g.) in 5 ml. dimethylformamide is then added and the mixture stirred for 24 hours at 110° under nitrogen. The resulting solution is poured into water (400 ml), extracted with ether (400 ml total), and the extracts washed, dried (MgSO4) and evaporated. The resulting crude solid (2.2 g) is recrystallized from toluene to give 1-[2-(2-naphthyl)-2,2-dimethoxyethyl]imidazole as a colorless solid.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04150153uspto-grants-1979_04