반응 #54592

ord-dc120655c6e54af49941a144e86ef0e0

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도This solution is heated
  2. 2
    온도is then refluxed for 5 minutes
  3. 3
    온도The mixture is refluxed for a further 2 minutes
  4. 4
    기타evaporated
  5. 5
    세척washed with water
  6. 6
    기타dried
  7. 7
    기타the solvent removed under vacuo

실험 절차

2-Aminopentanoic acid (0.2 mole) is added to a solution of sodium acetate (0.2 mole) in about 300 ml of glacial acetic acid. This solution is heated to effect solution and is then refluxed for 5 minutes. To the refluxing solution is added (0.2 mole) 2.5-dimethoxytetrahydrofuran as quickly as possible. The mixture is refluxed for a further 2 minutes and the acetic acid is flash evaporated. The residue is taken up in ethyl acetate, washed with water, dried and the solvent removed under vacuo to give 2-(1-pyrryl)pentanoic acid.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04148998uspto-grants-1979_04