반응 #54591

ord-238e2c7868bf4c0ab667f4ccfcc35579

반응 방정식

O
water
ClC(Cl)Cl
Chloroform
O=C1NC(=O)c2ccccc21.[K]
potassium phthalimide
CCCC(Br)C(=O)OCC
ethyl-2-bromopentanoate
CCCC(C(=O)OCC)N1C(=O)c2ccccc2C1=O
ethyl α-phthalimidopentanoate

반응 조건

온도
60°CELSIUS
상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타The phases are separated
  2. 2
    추출the aqueous phase is extracted with chloroform
  3. 3
    추출extracted with 0.1 N sodium hydroxide and with water
  4. 4
    건조After drying over sodium sulfate
  5. 5
    기타the chloroform is removed

실험 절차

To a solution of potassium phthalimide (0.1 mole) in about 50 ml of dimethylformamide (DMF) is added 1 equivalent of ethyl-2-bromopentanoate. The temperature is maintained at about 60° C. for 10 minutes. Chloroform is added to the cooled DMF solution and the mixture is poured into water. The phases are separated and the aqueous phase is extracted with chloroform. The chloroform extracts are combined, extracted with 0.1 N sodium hydroxide and with water. After drying over sodium sulfate, the chloroform is removed to give ethyl α-phthalimidopentanoate.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04148998uspto-grants-1979_04