반응 #526936

ord-22676dae95144dcb8920a1d205ec03c3

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도is cooled in an ice bath
  2. 2
    기타The solvent is removed under vacuum
  3. 3
    기타chromatographed on normal phase silica gel using a gradient from hexane to a 4:1 ratio of hexane

실험 절차

A mixture of 7.3 g of 60% NaH in 190 ml of anhydrous dimethylformamide is cooled in an ice bath. To this mixture is added 22.0 g of 3-pentyloxyphenol dissolved in 50 ml of anhydrous dimethylformamide. This mixture is then stirred at room temperature for 45 minutes; 23.2 ml of ethyl 4-bromobutyrate are added; and the resultant mixture is stirred at 60° C. for 17 hours. The solvent is removed under vacuum and the residue worked up as above. The residue is flash chromatographed on normal phase silica gel using a gradient from hexane to a 4:1 ratio of hexane:ether to yield ethyl 4-(3-pentyloxyphenoxy)butyrate as a clear oil.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05516767uspto-grants-1996_05