반응 #52658

ord-5e8a1e2bb0f9481c9e511871bbe592ce

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타the precipitate which formed
  2. 2
    여과was collected by vacuum filtration
  3. 3
    세척washed with 50 ml of water
  4. 4
    기타dried

실험 절차

A solution of 5-chloroacetyl-2-oxindole (4.18 g) in trifluoroacetic acid (30 ml) was cooled in an ice bath and 4.65 g of triethylsilane added. The mixture was then stirred at room temperature for 3 hours. The mixture was poured into 150 ml of water and the precipitate which formed was collected by vacuum filtration, washed with 50 ml of water and dried to give 2.53 g (65% yield) of 5-(2-chloroethyl)-2-oxindole as a reddish-brown solid.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US06855730B2uspto-grants-2005_02