반응 #51228

ord-3ec4e80e1edf430a8ee4eedd99c59306

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타Manganese dioxide was removed by filtration through Celite
  2. 2
    기타the solvent was removed under reduced pressure
  3. 3
    여과the crystals were collected by filtration

실험 절차

20 g of manganese dioxide was added to 120 ml of a chloroform solution containing 4.0 g of N-benzyloxycarbonyl-trans-4-[(5-hydroxymethyl-2-isoindolinyl)carbonyl]cyclohexylamine, and the mixture was stirred at room temperature for 4 hours. Manganese dioxide was removed by filtration through Celite and the solvent was removed under reduced pressure. The residue was suspended in hexane-ethyl acetate and the crystals were collected by filtration to obtain N-benzyloxycarbonyl-trans-4-[(5-formyl-2-isoindolinyl)carbonyl]cyclohexylamine.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US06849622B2uspto-grants-2005_02