반응 #50585

ord-4e9e7528c2ef4b708c884f4ab638ad29

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타Method A (23 h at 60° C.)

실험 절차

Method A (23 h at 60° C.); starting materials: 6-[3-(methanesulfonyloxy)propoxy]-7-methoxy-2H-1-benzopyran-2-one (see example 67) and 1-phenylpiperazine; yield 55%; fusion point 124° to 125° C. (from ethanol). Fumarate: method E; yield 88%; fusion point 172° to 173° C. (from ethanol).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05428038uspto-grants-1995_06