반응 #50129

ord-a0df9aa2b5d94cfb8738aba40dd8ebff

반응 조건

온도
140°CELSIUS
상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타A four-necked flask equipped with a gas inlet, a dry ice condenser, a mechanical stirrer
  2. 2
    기타to destroy traces of phosgene which
  3. 3
    기타condensed in the condenser
  4. 4
    기타to purge residual phosgene
  5. 5
    온도the reactor is cooled to ambient temperature
  6. 6
    기타The colorless crude product is isolated by vacuum distillation

실험 절차

A four-necked flask equipped with a gas inlet, a dry ice condenser, a mechanical stirrer, a thermocouple and a sampling port is charged with phenol (Aldrich, 287.5 g, 2.907 mol) and triphenyl phosphite (10.12 g, 32.61 mmol). The temperature is raised to 140° C. and phosgene (274 g, 2.77 mol) is added over a 465 minute period. Phosgene/phenol molar ratio is 0.95. A recirculating aqueous sodium hydroxide scrubber is used to neutralize the coproduct hydrochloric acid and to destroy traces of phosgene which are not condensed in the condenser. After the phosgene addition is stopped, a nitrogen stream is used to purge residual phosgene and the reactor is cooled to ambient temperature. The colorless crude product is isolated by vacuum distillation to give phenyl chloroformate (417.84 g, bp 73°-77° C. at 14 mm Hg) containing 6.6 percent by weight residual phenol. Selectivity to phenyl chloroformate is 95 mole percent based on phenol, 90 mole percent based on phosgene.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05424473uspto-grants-1995_06