반응 #48026

ord-580966e9b0a742c6aecadfce7399d1a3

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    추출The solution was extracted
  2. 2
    건조with water, 5% acetic acid and water, successively, dried over anh. sodium sulfate
  3. 3
    기타evaporated to dryness

실험 절차

14.7 g (52.8 mmol) of N-[2-hydroxy-3-(1-piperidinyl)propoxy]-3-pyridine-carboximidamide [Hung. Pat. 177.578 (1976)] was dissolved in 160 ml of chloroform. 7.7 ml (55 mmol) of triethylamine was added, followed by dropwise addition of a solution of palmitoyl chloride (14.7 g; 56.5 mmol) in 85 ml of chloroform. The mixture was stirred overnight at room temperature. Next day further amount of 3.8 ml of triethylamine and 7.4 g of palmitoylchloride was added, and the stirring was continued for one more day. The solution was extracted then with water, 5% acetic acid and water, successively, dried over anh. sodium sulfate, and evaporated to dryness.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US07745465B2uspto-grants-2010_06