반응 #477200

반응 방정식

3-amino-5,6-dihydro-6-N-(p-tolyl)-1H-pyrazolo[3,4-c]pyridin-7(4H)-one

potassium carbonate

3-chloro-1-{4-(4-methoxyphenyl)piperazin-1-yl}propan-1-one

→

3-amino-1-[{4-(4-methoxyphenyl)piperazin-1-yl}propanoyl]-6-N-(p-tolyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridin-7-one

반응 조건

실험 절차

A target compound (154.9 mg, 0.317 mmol, 76.9%) was yielded as white solid the same manner as in Example 1 by reacting 3-amino-5,6-dihydro-6-N-(p-tolyl)-1H-pyrazolo[3,4-c]pyridin-7(4H)-one (100 mg, 0.412 mmol) with potassium carbonate (85.4 mg, 0.618 mmol) and 3-chloro-1-{4-(4-methoxyphenyl)piperazin-1-yl}propan-1-one (128.1 mg, 0.453 mmol).

출처