반응 #46785

ord-be01ac0db92847d3925527deccc00814

용매

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    여과the mixture was filtered through a chem elut® cartridge by elution with ethyl acetate
  2. 2
    기타After removal of the solvent under reduced pressure the crude product
  3. 3
    기타was subjected to the next reaction step without further purification

실험 절차

To a solution of 300 mg 1H-Benzoimidazole-2-carboxylic acid in 3 mL DMF and 1 mL NEt3, 398 mg 1-Isopropyl-piperidin-4-ylamine hydrochloride and 470 mg BOP-Cl were added and the mixture was stirred for 3 h. Finally, 3 mL saturated NaHCO3 solution were added and the mixture was filtered through a chem elut® cartridge by elution with ethyl acetate. After removal of the solvent under reduced pressure the crude product was subjected to the next reaction step without further purification.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US07741341B2uspto-grants-2010_06