반응 #4537

ord-0e6c16dd3649420f8ec300810a013520

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    여과filtered over silica gel
  2. 2
    기타the filtrate was evaporated down

실험 절차

5.1 g of pyridinium chlorochromate were added a little at a time to a solution of 4 g of 3-hydroxymethyl-5-dichloromethyl-2-phthalimidopyrazine in 80 ml of dichloromethane at 35° C., after which the mixture was stirred for 40 minutes and filtered over silica gel, and the filtrate was evaporated down. 3.1 g (76%) of colorless crystals of 3-formyl-5-dichloromethyl-2-phthalimidopyrazine of melting point 145°-146° C. (from ethyl acetate) were obtained. 1H-NMR (270 MHz, CDCl3): δ6.9 (s, 1H), 8.0 (m, 4H), 9.3 (s, 1H), 10.1 (s, 1H).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04725689uspto-grants-1988_02