반응 #4287

ord-cc9151e5ad6b4f33b85396bdbeeebe64

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도with cooling in an ice bath
  2. 2
    여과filtered
  3. 3
    기타Solvent was removed from the filtrate in a rotary evaporator
  4. 4
    기타to give an oil which
  5. 5
    기타crystallized
  6. 6
    기타A portion was recrystallized from isopropyl ether
  7. 7
    기타to give white crystalline solid, m.p. 53°-55° C.

실험 절차

To a solution of 117.97 g (0.53 mole) of 2-[(3,4-dichlorophenyl)thio]ethanol (prepared by reacting 3,4-dichlorothiophenol and 2-chloroethanol) and 53.5 g (0.53 mole) of triethylamine in 500 ml of benzene was added dropwise a benzene solution of 60.9 g (0.53 mole) of methanesulfonyl chloride over a one hour period with cooling in an ice bath. The reaction mixture was stirred at room temperature overnight and filtered. Solvent was removed from the filtrate in a rotary evaporator to give an oil which crystallized. A portion was recrystallized from isopropyl ether to give white crystalline solid, m.p. 53°-55° C.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US04724235uspto-grants-1988_02