반응 #3142

ord-4d14267579d347aaab5da8765031fa8d

반응 방정식

CC1(N)N=C(O)C=C(O)N1
4,6-dihydroxy-2-methylpyrimidinamine
CC[O-].[Na+]
sodium ethoxide
[Na]
sodium
CC(=N)N.Cl
Acetamidine hydrochloride
CCOC(=O)CC(=O)OCC
diethyl malonate
Cc1nc(O)cc(O)n1
4,6-dihydroxy-2-methylpyrimidine

용매

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도the reaction mixture heated

실험 절차

The first intermediate, 4,6-dihydroxy-2-methylpyrimidinamine, is synthesized by preparing sodium ethoxide in situ from sodium and an hydrous ethanol under a nitrogen blanket. Acetamidine hydrochloride and diethyl malonate are added and the reaction mixture heated to boiling for 2 to 5 hours to afford 4,6-dihydroxy-2-methylpyrimidine.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05732717uspto-grants-1998_03