반응 #217506

ord-20bbbca9340448099b93274c4af3fd17

반응 조건

온도
100°CELSIUS
상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타A vigorous exothermic reaction
  2. 2
    여과The solid was filtered
  3. 3
    세척washed with water
  4. 4
    기타dried

실험 절차

To a heated mixture (in an oversized flask) of 13 g (63 mmol) 4,6-dimethoxyindole-2,3-dione prepared in Example 1 and 108 ml of 33% NaOH solution was carefully added 20 ml of a 30% solution of H2O2. A vigorous exothermic reaction occurs. After all H2O2 was added, the reaction mixture was maintained at 100° C. for an additional 10 min. The pH of the solution was brought to 8 with concentrated HCl and acidified to pH 5-6 with acetic acid. The solid was filtered, washed with water and dried to yield 6.2 g of 4,6-dimethoxyanthranilic acid as a pale brown solid (50% yield).

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US07381730B2uspto-grants-2008_06