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[7-(2-{[tert-butyl(dimethyl)silyl]oxy}-1,1-dimethylethyl)-2-amino-7H-pyrrolo[2,3-d]pyrimidin-5-yl]{5-aminopyridin-3-yl}methanone

[4-(trifluoromethyl)-1H-1,2,3-triazol-1-yl]acetic acid

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title compound

N-(5-{[2-Amino-7-(2-hydroxy-1,1-dimethylethyl)-7H-pyrrolo[2,3-d]pyrimidin-5-yl]carbonyl}pyridin-3-yl)-2-[4-(trifluoromethyl)-1H-1,2,3-triazol-1-yl]acetamide

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후처리

1. 1
   기타The title compound was prepared

실험 절차

The title compound was prepared according to the method described for Example 9 using [7-(2-{[tert-butyl(dimethyl)silyl]oxy}-1,1-dimethylethyl)-2-amino-7H-pyrrolo[2,3-d]pyrimidin-5-yl]{5-aminopyridin-3-yl}methanone (see Preparation 48a) and [4-(trifluoromethyl)-1H-1,2,3-triazol-1-yl]acetic acid (see Preparation 81) to afford the title compound as a brown solid in 85% yield, 62 mg.

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