반응 #157922

ord-7c2b84a7b779425e99164e43cf496820

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    세척The organic phase was washed with saturated NaHCO3 (3×10 mL), dried Na2SO4
  2. 2
    농축concentrated in vacuo

실험 절차

Phenyl cyclohexene (50 mg) and thiophene (100 mg) were dissolved in 33% HBr in acetic acid (0.5 mL). The mixture was stirred at room temperature over night. Tlc indicated full conversion of the starting material. Dichloromethane (10 mL) was added. The organic phase was washed with saturated NaHCO3 (3×10 mL), dried Na2SO4 and concentrated in vacuo. The desired product was afforded after flash chromatography (eluent: dichloromethane). Yield: 39 mg. LC/MS purity (UV/MS): 100/90%, Rt 6.22 min. M+1: 243

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US08822548B2uspto-grants-2014_09