반응 #1502

ord-169f88b27a294c15b3d94e8de0e682c6

반응 방정식

O=C(Cl)OCCl
Chloromethyl chloroformate
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@@H](O)CC[C@]4(C)[C@H]3CC[C@]12C
cholesterol
c1ccncc1
Pyridine
CC(C)CCC[C@@H](C)[C@H]1CC[C@H]2[C@@H]3CC=C4C[C@](O)(C(=O)OCCl)CC[C@]4(C)[C@H]3CC[C@]12C
3-(Chloromethoxycarbonyl) Cholesterol

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    온도The solution was cooled
  2. 2
    온도Heat
  3. 3
    기타was produced
  4. 4
    기타the reaction gave a clear solution from
  5. 5
    세척washed with 0.5M HCl (50 ml) and water (3×25 ml)
  6. 6
    기타After treatment with MgSO4, the solution was evaporated to dryness

실험 절차

Chloromethyl chloroformate (1.96 g, 15.2 mmol) and cholesterol (5.0 g, 12.9 mmol) was dissolved in CH2Cl2 (10 ml). The solution was cooled. Pyridine (1.21 g, 15.3 mmol) was dripped into the stirred solution over 5 minutes. Heat was produced and the reaction gave a clear solution from a somewhat unclear starting solution. After 24 hours at room temperature, the mixture was diluted with CH2Cl2 (50 ml), washed with 0.5M HCl (50 ml) and water (3×25 ml). After treatment with MgSO4, the solution was evaporated to dryness.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US05725840uspto-grants-1998_03