반응 #12059

ord-1c7e89d4d4514972a067ddc65a248326

반응 조건

상세 조건
See reaction.notes.procedure_details.

후처리

  1. 1
    기타This was capped with a Dean-Stark trap
  2. 2
    온도heated
  3. 3
    온도to reflux for two hours at which time the system
  4. 4
    기타the volatiles removed in vacuo
  5. 5
    기타to leave a dark oil
  6. 6
    세척eluted through a silica pad
  7. 7
    기타Removal of the volatiles in vacuo

실험 절차

A 500 mL flask was charged with 25.5 g (120 mmol) of trans-2-bromo-1-indanol, 1 g of toluenesulfonic acid and 350 mL of toluene. This was capped with a Dean-Stark trap and heated to reflux for two hours at which time the system was cooled to room temperature and the volatiles removed in vacuo to leave a dark oil. The residue was taken up into hexanes and eluted through a silica pad using hexanes. Removal of the volatiles in vacuo gave 22.5 g (96 percent) of a light yellow oil.

출처

DOI: 10.6084/m9.figshare.5104873.v1특허: US07098356B2uspto-grants-2006_08