반응 #1114168

반응 방정식

7-chloro-3-ethoxycarbonyl-6-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidine

7-Chloro-3-ethoxycarbonyl-6-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidine

1-methyl-5-aminoindole

→

title compound

수율 90.0%

3-Ethoxycarbonyl-7-(1-methyl-5-indolylamino)-6-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidine

수율 90.0%

반응 조건

실험 절차

In the same manner as in Example 19, step 5 and using 7-chloro-3-ethoxycarbonyl-6-(4-phenylpiperidine-1-carbonyl)pyrazolo[1,5-a]pyrimidine (0.15 g, 0.36 mmol) obtained in Example 19, step 4 and 1-methyl-5-aminoindole (0.072 g, 0.49 mmol), the title compound (0.169 g, 90%) was obtained.

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