反応 #68797

反応方程式

(S)-[1-(4-Bromo-phenyl)-ethyl]-carbamic acid tert-butyl ester

(S)-[1-(4-bromo-phenyl)-ethyl]-carbamic acid tert-butyl ester

3-(4-cyclopropylmethoxy-phenoxy)-azetidine

→

(S)-(1-{4-[3-(4-Cyclopropylmethoxy-phenoxy)-azetidin-1-yl]-phenyl}-ethyl)-carbamic acid tert-butyl ester

反応条件

後処理

1. 1
   その他Example 8.3 is prepared analogously to 8.1
2. 2
   その他is 45° C.

実験手順

Example 8.3 is prepared analogously to 8.1. (S)-[1-(4-Bromo-phenyl)-ethyl]-carbamic acid tert-butyl ester (1.3) and 3-(4-cyclopropylmethoxy-phenoxy)-azetidine (IX.1) are used as starting materials and the reaction temperature is 45° C.

出典