反応 #60810

ord-bfa91bba01444c858e262522dcf3c6d5

反応方程式

C[S-].[Na+]
sodium thiomethoxide
Cc1cc2ncnc(Cl)c2s1
6-methyl-4-chlorothieno[3,2-d]pyrimidine
CSc1ncnc2cc(C)sc12
title compound
収率 97.0%
CSc1ncnc2cc(C)sc12
6-Methyl-4-(methylthio)thieno[3,2-d]pyrimidine
収率 97.0%

反応条件

詳細条件
See reaction.notes.procedure_details.

後処理

  1. 1
    ろ過The mixture was filtered
  2. 2
    洗浄the solid was washed with acetonitrile
  3. 3
    その他The combined filtrate and washes were evaporated

実験手順

A solution of sodium thiomethoxide (24S mg) and 6-methyl-4-chlorothieno[3,2-d]pyrimidine (Acta Pol. Pharm. (1986), 43(2), 97-100) (650 mg) in acetonitrile (50 mL) was stirred overnight. The mixture was filtered and the solid was washed with acetonitrile. The combined filtrate and washes were evaporated to give the title compound as a white solid (665 mg, 97%);

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US07427616B2uspto-grants-2008_09