反応 #430112

ord-a287f31b9303459e8fd267ab8b600b01

反応条件

詳細条件
See reaction.notes.procedure_details.

実験手順

It has been found that, surprisingly, when neutralizing (S)-2-(6-methoxy-2-naphthyl)propionic acid having a chiral purity below 99% with less than a stoichiometric amount of aqueous sodium hydroxide solution to form naproxen sodium, it is possible to increase the chiral purity of the naproxen sodium to 99% or more by removing the water by use of a suitable organic solvent, or simply by distilling off water from an aqueous solution.

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US05859292uspto-grants-1999_01