反応 #41331

ord-e34e34bb15ff4c30886fee6ddbb92d8e

反応条件

詳細条件
See reaction.notes.procedure_details.

後処理

  1. 1
    その他Prepared

実験手順

Prepared as described in Example 1 using (1R,2S)-1-(4-ethylphenyl)-1-{[1-(4-fluorophenyl)-1H-indazol-5-yl]oxy}propan-2-amine (7a, 20 mg, 50 μmol) and 2-methylpropanoyl chloride (16 mg, 150 nmol). Yield 18 mg (78%).

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US07728030B2uspto-grants-2010_06