反応 #41319

ord-8b46b6b3e5434be69719c72453e58e27

反応条件

詳細条件
See reaction.notes.procedure_details.

後処理

  1. 1
    その他Prepared

実験手順

Prepared as described in Example 1 using (1S,2R)-1-{[1-(4-fluorophenyl)-1H-indazol-5-yl]oxy}-1-phenylpropan-2-amine (1a, 18 mg, 50 μmol) and 2-methylpropanoyl chloride (21 mg, 150 μmol). Yield 18 mg (84%).

出典

DOI: 10.6084/m9.figshare.5104873.v1特許: US07728030B2uspto-grants-2010_06